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CALCIMIMETIC AGENTS
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DeCS
Descriptor
English
:
Calcimimetic Agents
Descriptor
Spanish
:
Agentes Calcimiméticos
Descriptor
Portuguese
:
Calcimiméticos
Tree Number:
D06.347.230
D27.505.696.399.450.230
Definition
English
:
Small organic molecules that act as allosteric activators of the
calcium
sensing receptor (CaSR) in the
PARATHYROID GLANDS
and other
tissues
. They lower the threshold for CaSR activation by extracellular
calcium
ions
and diminish
PARATHYROID HORMONE
(PTH) release from parathyroid
cells.
History Note
English
:
2011
Allowable Qualifiers
English
:
AD
administration & dosage
AE
adverse effects
AG
agonists
AN
analysis
BL
blood
CF
cerebrospinal fluid
CS
chemical synthesis
CH
chemistry
CL
classification
CT
contraindications
DU
diagnostic use
EC
economics
HI
history
IM
immunology
IP
isolation & purification
ME
metabolism
PK
pharmacokinetics
PD
pharmacology
PO
poisoning
RE
radiation effects
ST
standards
SD
supply & distribution
TU
therapeutic use
TO
toxicity
UR
urine
Record Number:
54038
Unique Identifier:
D057966
Occurrence in VHL
:
Similar:
DeCS
CID-10
SciELO
LILACS
LIS